Lead Generation Approaches in Drug Discovery H 308 p. 10
Rankovic, Z 著
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PREFACE. CONTRIBUTORS. 1 Lead Discovery: The Process (William F. Michne). 2 High Throughput Screening Approach to Lead Discovery (Zoran Rankovic, Craig Jamieson, and Richard Morphy). 3 In Silico Screening (Dagmar Stumpfe, Hanna Geppert, and Jürgen Bajorath). 4 Fragment–Based Lead Discovery (Jeffrey S. Albert). 5 Design of Multitarget Ligands (Richard Morphy and Zoran Rankovic). 6 De novo Drug Design (Gisbert Schneider, Markus Hartenfeller, and Ewgenij Proschak). 7 Role of Natural Products in Drug Discovery (Hugo Lachance, Stefan Wetzel, and Herbert Waldmann). 8 Early Screening for ADMET Properties (Dennis A. Smith). 9 Role of Chemistry in Lead Discovery (Roland E. Dolle and Karin Worm). INDEX.
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